Description
An alpha, beta-Methylene-ADP (AOPCP) derivative, potent, selective ecto-5'-Nucleotidase (eN, CD73) inhibitor with Ki of 29nM for rat recombinant eN; also exhibits dual-action properties toward both A2AR and equilibrative nucleoside transporter 1 (ENT1) with Ki of 27.7uM and 6.51nM